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dc.contributor.author | Rodríguez Agudo, Rubén | |
dc.contributor.author | Petrov, Petar D. | |
dc.contributor.author | Castell, José V. | |
dc.contributor.author | over Atienza, Ramiro | |
dc.date.accessioned | 2023-05-29T13:33:09Z | |
dc.date.available | 2023-05-29T13:33:09Z | |
dc.date.issued | 2022 | |
dc.identifier.citation | Rodríguez Agudo, Rubén Petrov, Petar D. Castell, José V. over Atienza, Ramiro 2022 Methionine cycle rewiring by targeting miR-873-5p modulates ammonia metabolism to protect the liver from acetaminophen Antioxidants 11 5 897 | |
dc.identifier.uri | https://hdl.handle.net/10550/87070 | |
dc.description.abstract | Drug-induced liver injury (DILI) development is commonly associated with acetaminophen (APAP) overdose, where glutathione scavenging leads to mitochondrial dysfunction and hepatocyte death. DILI is a severe disorder without effective late-stage treatment, since N-acetyl cysteine must be administered 8 h after overdose to be efficient. Ammonia homeostasis is altered during liver diseases and, during DILI, it is accompanied by decreased glycine N-methyltransferase (GNMT) expression and S-adenosylmethionine (AdoMet) levels that suggest a reduced methionine cycle. Anti-miR-873-5p treatment prevents cell death in primary hepatocytes and the appearance of necrotic areas in liver from APAP-administered mice. In our study, we demonstrate a GNMT and methionine cycle activity restoration by the anti-miR-873-5p that reduces mitochondrial dysfunction and oxidative stress. The lack of hyperammoniemia caused by the therapy results in a decreased urea cycle, enhancing the synthesis of polyamines from ornithine and AdoMet and thus impacting the observed recovery of mitochondria and hepatocyte proliferation for regeneration. In summary, anti-miR-873-5p appears to be an effective therapy against APAP-induced liver injury, where the restoration of GNMT and the methionine cycle may prevent mitochondrial dysfunction while activating hepatocyte proliferative response. | |
dc.language.iso | eng | |
dc.relation.ispartof | Antioxidants, 2022, vol. 11, num. 5, p. 897 | |
dc.subject | Bioquímica clínica | |
dc.title | Methionine cycle rewiring by targeting miR-873-5p modulates ammonia metabolism to protect the liver from acetaminophen | |
dc.type | journal article | |
dc.date.updated | 2023-05-29T13:33:09Z | |
dc.identifier.doi | 10.3390/antiox11050897 | |
dc.identifier.idgrec | 159246 | |
dc.rights.accessRights | open access |